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Arenes

Reactions

Electrophilic Substitution

\(\require{mhchem}\ce{Benzene + Cl_2 -> Chlorobenzene + Cl^-}\) \(NO_2\ ^+\) can be replaced with any other electrophile (e.g. \(^+CH_3\))

Side-chain substitution

Same as alkane

Substituents

\(e^-\) withdrawing \(e^+\) donating \(-X\) groups
AKA Deactivating Groups Activating Groups Activating
Example Groups \(-COOH\), \(-COOR\), \(-C≡N\), \(-CONR\) \(-R\), \(-OR\), \(-OH\), \(-NR_2\) \(-Cl\), \(-Br\)
Features Unsaturated Saturated Saturated
Rate of rxn Decreased Increased Increased
Why? Decreased electron density, less susceptible to electrophilic attacks Increased electron density, more susceptible to electrophilic attacks Backdonation
Directing Positions 1, 3, 5 2, 4, 6 1, 3, 5